Contents

Noah Burns
(Columbia University)
Currently: Assistant Professor, Stanford University
Currently: Assistant Professor, Stanford University

Michael DeMartino
(University of Delaware)
Currently: GlaxoSmithKline
Currently: GlaxoSmithKline

Carlos Guerrero
(Harvard University)
Currently: Bristol-Myers Squibb
Currently: Bristol-Myers Squibb

Ben Hafensteiner
(University of Rochester)
Currently: Instructor, Rochester University
Currently: Instructor, Rochester University

Yoshihiro Ishihara
(McGill University)
Currently: Vertex Pharmaceuticals
Currently: Vertex Pharmaceuticals

Paul Krawczuk
(New York University)
Currently: Johnson & Johnson
Currently: Johnson & Johnson

David Lin
(Stanford University)
Currently: Johnson & Johnson
Currently: Johnson & Johnson

Jonathan Lockner
(University of Illinois at Urbana-Champaign)
Currently: Chair ACS San Diego
Currently: Chair ACS San Diego

Dan O'Malley
(Rice University)
Currently: Bristol-Myers Squibb
Currently: Bristol-Myers Squibb

Tim Newhouse
(Colby College)
Currently: Assistant Professor, Yale University
Currently: Assistant Professor, Yale University

Jeremy Richter
(Butler University)
Currently: Bristol-Myers Squibb
Currently: Bristol-Myers Squibb

Tom Maimone
(University of California, Berkeley)
Currently: Assistant Professor, University of California, Berkeley
Currently: Assistant Professor, University of California, Berkeley

Ian Seiple
(University of California, Berkeley)
Currently: Assistant Professor, University of California San Francisco
Currently: Assistant Professor, University of California San Francisco

Ryan Shenvi
(Penn State University)
Currently: Associate Professor, The Scripps Research Institute
Currently: Associate Professor, The Scripps Research Institute

Jun Shi
(Wuhan University, China)
Currently: Bristol-Myers Squibb
Currently: Bristol-Myers Squibb

Ana-Florina Voica
(Smith College)
Currently: Gilead
Currently: Gilead

Hans Renata
(Columbia University)
Currently: Assistant Professor, Scripps Florida
Currently: Assistant Professor, Scripps Florida

Will Gutekunst,
(University of Oklahoma)
Currently: Assistant Professor, Georgia Tech
Currently: Assistant Professor, Georgia Tech

Klement Foo
(Imperial College London)
Currently: A*STAR Research Center
Currently: A*STAR Research Center

Emily Cherney
(The College of New Jersey)
Currently: Bristol-Myers Squibb
Currently: Bristol-Myers Squibb

Steve McKerrall
(University of Maryland, Baltimore)
Currently: Genentech
Currently: Genentech

Dane Holte
(Northwestern University)
Currently: Stemcentrx
Currently: Stemcentrx

Rodrigo Rodriguez
(San Diego State University)
Currently: GNF
Currently: GNF

Quentin Michaudel
(École Normale Supérieure de Lyon)
Currently: Postdoctoral Associate Brett Fors
Currently: Postdoctoral Associate Brett Fors

Ryan Gianatassio
Currently: Biogen

Brandon Rosen
(University of Michigan)
Currently: Arcus Biosciences
Currently: Arcus Biosciences

Nathan Wilde
(Brigham Young University)
Currently: Postdoctoral Associate E. J. Corey
Currently: Postdoctoral Associate E. J. Corey

Leah Simke
(University of Michigan)
Currently: Pharmaron
Currently: Pharmaron

Hai Dao
Currently: Postdoctoral Associate Tom Muir

Matt Villaume
Currently: Vanderbilt University School of Medicine

Artiom Cernijenko
(Oxford University)
Currently: Novartis
Currently: Novartis

Julian Lo
(University of Minnesota)
Currently: Bristol-Myers Squibb
Currently: Bristol-Myers Squibb

Ruben Martinez
(University Of California Urvine)
Currently: IDEAYA Pharma
Currently: IDEAYA Pharma

Ming Yan
(LaFayette College)
Currently: Fish & Richardson
Currently: Fish & Richardson

Marcus Farmer
(University of South Florida)
Currently: Postdoctoral Associate Paul Chirik
Currently: Postdoctoral Associate Paul Chirik

Hang Chu
(University of Chicago)
Currently: Gilead
Currently: Gilead

Jacob Edwards
(University of Minnesota)
Currently: Celgene
Currently: Celgene

Yi Yang See
(University of Cambridge)
Currently: Postdoctoral Associate Melanie Sanford
Currently: Postdoctoral Associate Melanie Sanford

Justine deGruyter
(New Mexico State University)
Currently: Fish & Richardson
Currently: Fish & Richardson

Rohan Merchant
(University College London)
Merck
Merck

Yuzuru Kanda
(University of Tokyo)
Currently: Postdoctoral Associate in Radosevich Lab (MIT)
Currently: Postdoctoral Associate in Radosevich Lab (MIT)

Solomon Reisberg
(Kenyon College)
Currently: Third Rock Ventures
Currently: Third Rock Ventures

Thomas Stratton
(Rutgers University)
Currently: Gilead
Currently: Gilead

Kyle McClymont
(University of Ottawa)
Currently: Merck
Currently: Merck

Lisa Barton
(Northeastern University)
Currently: Genentech
Currently: Genentech

Kyle Knouse
(Temple University)
Currently: Co-Founder at Elsie Biotechnologies
Currently: Co-Founder at Elsie Biotechnologies

David Peters
(USD)
Currently: BMS
Currently: BMS

Jieyu Gu
(Peking University of Health Science Center)

Stephen Harwood
(UC Berkeley)
Currently: Mirati Therapeutics
Currently: Mirati Therapeutics

Maximilian Palkowitz
(Boston College)
Currently: Bristol Myers Squibb
Currently: Bristol Myers Squibb
Postdoctoral Associates

Alexandros Zografos
(National Technical University of Athens)
Currently: Aristotle University of Thessaloniki
Currently: Aristotle University of Thessaloniki

Ian Young
(University of Western Ontario)
Currently: Bristol-Myers Squibb
Currently: Bristol-Myers Squibb

Karin Weidner
(University of Bern)
Currently: Postdoctoral Associate Masakatsu Shibasaki
Currently: Postdoctoral Associate Masakatsu Shibasaki

Junichiro Yamaguchi
(Tokyo University of Science)
Currently: Associate Professor, Nagoya University
Currently: Associate Professor, Nagoya University

Ippei Usui
(Albert-Ludwigs-Universität Freiburg)
Currently: Sirenas Marine Discovery
Currently: Sirenas Marine Discovery

Andreas Weickgenannt
(Westfälische Wilhelms– Universität Münster)
Currently: BASF
Currently: BASF

Shun Su
(Boston University)
Currently: Bristol-Myers Squibb
Currently: Bristol-Myers Squibb

Damien Thevenet
(University of Neuchâtel)
Currently: Postdoctoral Associate Reinhard Neier
Currently: Postdoctoral Associate Reinhard Neier

Niklas Schöne
(Universität Stuttgart)
Currently: Sandoz, Austria
Currently: Sandoz, Austria

Hiroki Shigehisa
(Hoshi University)
Currently: Assistant Professor, Musashino University
Currently: Assistant Professor, Musashino University

Masanori Nagatomo
(The University of Tokyo)
Currently: Assistant Professor, The University of Tokyo
Currently: Assistant Professor, The University of Tokyo

Elena Petricci
(Università degli Studi di Siena)
Currently: Università degli Studi di Siena, Italy
Currently: Università degli Studi di Siena, Italy

Michael Maue
(Philipps-Universtität Marburg)
Currently: Bayer CropScience
Currently: Bayer CropScience

Abraham Mendoza
(University of Oviedo)
Currently: Assistant Professor, Stockholm University
Currently: Assistant Professor, Stockholm University

Georg Manolikakes
(Ludwig-Maximilians-Universität München)
Currently: Geothe Universität, Frankfurt am Main
Currently: Geothe Universität, Frankfurt am Main

Takeshi Masuda
(University of Tokyo)
Currently: Daiichi-Sankyo Co., Ltd.
Currently: Daiichi-Sankyo Co., Ltd.

Ke Li
(New York University)
Currently: DuPont
Currently: DuPont

Mike Luzung
(University of California, Berkeley)
Currently: Bristol-Myers Squibb
Currently: Bristol-Myers Squibb

Chad Lewis
(Yale University)
Currently: Pfizer
Currently: Pfizer

Chuang Chuang Li
(Peking University, China)

Tanja Gulder
(University of Würzburg)
Currently: Research Group Leader, Technische Universität München
Currently: Research Group Leader, Technische Universität München

Mikkel Jessing
(Technical University of Denmark)
Currently: H. Lundbeck A/S
Currently: H. Lundbeck A/S

Yuta Fujiwara
(Gifu Pharmaceutical University)
Currently: Meiji Seika Pharma Co., Ldt.
Currently: Meiji Seika Pharma Co., Ldt.

Daniel Götz
(University of Würzburg)
Currently: Bayer, Wuppertal
Currently: Bayer, Wuppertal

Kyle Eastman
(Penn State University)
Currently: Bristol-Myers Squibb
Currently: Bristol-Myers Squibb

Tanja Gaich
(University of Vienna)
Currently: Assistant Professor, Leibniz Universität Hannover
Currently: Assistant Professor, Leibniz Universität Hannover

Ke Chen
(University of Rochester)
Currently: Bristol-Myers Squibb
Currently: Bristol-Myers Squibb

Darryl Dixon
(University of Hawaii at Manoa)
Currently: Bristol-Myers Squibb
Currently: Bristol-Myers Squibb

Moritz Biskup
(Universität Konstanz)
Currently: Karlsruher Institut für Technologie
Currently: Karlsruher Institut für Technologie

Tobias Brückl
(Ludwig-Maximilians-Universität München)
Currently: Merck Serano
Currently: Merck Serano

Narendra Ambhaikar
(Emory University)
Currently: TEVA Pharmaceuticals
Currently: TEVA Pharmaceuticals

Shinji Ashida
(Kyoto University)
Currently: Daiichi-Sankyo Co., Ltd.
Currently: Daiichi-Sankyo Co., Ltd.

Jason Green
(University of California, Santa Barbara)
Currently: Takeda San Diego
Currently: Takeda San Diego

Guillaume Journot
(University of Neuchâtel)
Currently: University of Munich
Currently: University of Munich

Lars Joergensen
(University of Copenhagen)
Currently: LEO Pharma
Currently: LEO Pharma

Christian Kuttruff
(Ludwig-Maximilians-Universität München)
Currently: Boehringer Ingelheim
Currently: Boehringer Ingelheim

Fionn O'Hara
(University of Cambridge)
Currently: Roche
Currently: Roche

Minetaka Isomura
(The University of Tokyo)
Currently: Eisai Co., Ltd.
Currently: Eisai Co., Ltd.

Erik Werner
(University of Utah)
Currently: Gilead Sciences
Currently: Gilead Sciences

Insa Prochnow
(University of Oldenburg)

Sarah Wengryniuk
(Duke University)
Currently: Assistant Professor, Temple University
Currently: Assistant Professor, Temple University

Akinobu Maruyama
(Osaka University)
Currently: Teijin Pharma. Limited
Currently: Teijin Pharma. Limited

Yuki Yabe
(Gifu Pharmaceutical University)
Currently: Eisai
Currently: Eisai

Bart Roman
(Ghent University)
Currently: Ghent University
Currently: Ghent University

Rune Risgaard
(University of Copenhagen)
Currently: LEO Pharma
Currently: LEO Pharma

Isabelle Thome
(RWTH Aachen University)
Currently: Roche
Currently: Roche

Qianghui Zhou
Currently: Professor, Wuhan University

Chien-Hung Yeh
(National Tsing Hua University)
Currently: TSRI
Currently: TSRI

Myles Smith
(Columbia University)
Currently: Stanford
Currently: Stanford

Ying Jin
Currently: Professor, Jilin Medical College

Eran Sella
Currently: Teva Pharmaceutical Industries

Kevin Oberg
(Colorado State University)
Currently: Eli Lilly
Currently: Eli Lilly

Yehua Jin

Changxia Yuan
Currently: Bristol-Myers Squibb

Jinghan Gui
(SIOC)
Currently: Professor, SIOC
Currently: Professor, SIOC

Shuhei Kawamura
(Hokkaido University)
Currently: Merck
Currently: Merck

Yu Feng
Currently: Abide Therapeutics

Chung-Mao Pan
(San Diego State University)
Currently: Sirenas Marine Discovery
Currently: Sirenas Marine Discovery

Fumihiko Toriyama
Currently: Daiichisankyo Co., Ltd.

Evan Horn
(University of California, Urvine)
Currently: Celgene
Currently: Celgene

Shigenobu Umemiya
(Tohoku University)
Currently: Assistant Professor, Tohoku University
Currently: Assistant Professor, Tohoku University

Maoqun Tian
Currently: Merck

Josep Cornella
(Queen Mary University of London)
Currently: Professor, Max Planck
Currently: Professor, Max Planck

Justin M. Lopchuk
(Dartmouth)
Currently: Assistant Professor, Moffitt Cancer Center
Currently: Assistant Professor, Moffitt Cancer Center

Aaron Herrmann
(University of California, Santa Barbra)
Currently: Janssen Pharmaceuticals
Currently: Janssen Pharmaceuticals

Koji Kobayashi
Currently: Astellas Pharmaceuticals

Lara Malins
(The University of Sydney)
Currently: Assistant Professor Australia National University
Currently: Assistant Professor Australia National University

Laurin Wimmer
(Vienna University of Technology)
Currently: Novartis
Currently: Novartis

Chao Li
(National Institute of Biological Sciences, Beijing)
Currently: Assistant Professor, National Institute of Biological Sciences, Beijing
Currently: Assistant Professor, National Institute of Biological Sciences, Beijing

Mayumi Yamaguchi

Joel Smith
(UCLA)
Currently: Assistant Professor, Florida State University
Currently: Assistant Professor, Florida State University

Javier Lopez Ogalla

Tian Qin
(Boston University)
Currently: Assistant Professor, UT Southwestern
Currently: Assistant Professor, UT Southwestern

Chuanguan Qin
Northwestern Polytechnical University

Karla Feu
The University of Campinas

Jie Wang
SIOC
Currently: Calibr
Currently: Calibr

David Kossler
École polytechnique fédérale de Lausanne

Shota Asai
Gifu Pharmaceutical University
Currently: Iwate University
Currently: Iwate University

Pavel Mykhailiuk
Enamine Ltd

Jinbao Xiang
Jilin University

Massimiliano Lamberto
Monmouth University

Xuejing Zhang
Sun Yat-sen University

Cian Kingston
(University College Dublin)
Currently: Postdoctoral Associate at The University of Utah with Matt Sigman
Currently: Postdoctoral Associate at The University of Utah with Matt Sigman

Tie-Gen Chen
SIOC

Yusuke Takahira
AGC Asahi Glass

Johannes Teske
University of Stuttgart

Byron Peters
(Stockholm University)
Currently: Merck
Currently: Merck

Natalia Muñoz Padial
Currently: University of Granada

Ming Shang
(SIOC)
Currently: Assistant Professor at SJTU
Currently: Assistant Professor at SJTU

Julien Vantourout
(University of Strathclyde)
Currently: Assistant Professor at CNRS (Centre national de la recherche scientifique)
Currently: Assistant Professor at CNRS (Centre national de la recherche scientifique)

Gary Hermann
(RTWH Aachen University)
Currently: Bayer
Currently: Bayer

Pengfei Hu
(University of Chicago)
Currently: Assistant Professor at Westlake University
Currently: Assistant Professor at Westlake University

Cody Pitts
(Johns Hopkins University)
Currently: Assistant Professor, UC Davis
Currently: Assistant Professor, UC Davis

Hugh Nakamura
(Kyoto University)
Currently: Assistant Professor, The Hong Kong University of Science and Technology
Currently: Assistant Professor, The Hong Kong University of Science and Technology

Kevin Rodriguez
(University of Notre Dame)
Currently: Gilead
Currently: Gilead

Michael Meanwell
Currently: University of Alberta

Chi He
Currently: BMS

Kyohei Hayashi
Currently: PLEXIUM

Adriano Bauer
(University of Vienna)
Currently: Amgen
Currently: Amgen

Jin Choi
(Seoul National University)
Currently: Odyssey Therapeutics
Currently: Odyssey Therapeutics

Samer Gnaim
(Tel-Aviv University)
Currently: Assistant Professor at Weizmann Institute of Science
Currently: Assistant Professor at Weizmann Institute of Science

Debora Chiodi
(University of Pavia)
Currently: Takeda Pharmaceuticals
Currently: Takeda Pharmaceuticals

Terry Lou
(University of Oxford)
Currently: Octant
Currently: Octant
Visiting Graduate Students

Jessica Giacoboni
University of Copenhagen-Lundbeck

Liher Prieto
University of the Basque Country

Chien-Hung Yeh
National Tsing Hua University

Jose Antonio Romero Revilla
Autonoma University of Madrid

Roy Weinstein
Tel Aviv University, Israel

Takeshi Yasui
Nagoya University

Felix Ungeheuer
University of Frankfurt

Tatsuya Urushima
Tokyo University of Science

Eran Sella
Tel Aviv University, Israel

Julian Shaw
Trinity College, Dublin

Amit Sagi
Tel Aviv University, Israel

Mariá Escribano Santamarina
Universidad De Oviedo, Spain

Rune Risgaard
University of Copenhagen

Alessandro Ruffoni
University of Milan D.I.S.F.A.R.M.

Akifumi Nakamura
The University of Tokyo

Antti Pohjakallio
Teknillinen Korkeakoulu-Helsinki University of Technology, Finland

Tomás Llamas
Universidad Autónoma de Madrid, Spain

Quentin Michaudel
École Normale Supérieure de Lyon

Yi Ning Ji Chen
Science Park of Barcelona

Lars Joergensen
University of Copenhagen

Kentaro Iso
Tohoku University

Mikkel Jessing
Technical University of Denmark

Cornelius Gropp
University of Heidelberg

Bart Herle
University of Amsterdam

Jorge Otero Fraga
University of Santiago de Compostela

Mariá Morón Galán
Universidad De Alcalá, Spain

Johan Dam
Technical University of Denmark

Victoriano Domingo
University of Granada

Pilar Castroviejo
Universidad de Burgos, Spain

Erik Daa Funder
University of Aarhus

César Rogelio Solorio Alvarado
Institute of Chemical Research of Catalonya

Ivan Bernar
UpSolution Team
Freie Universität Berlin

Marta Artola
Universidad Complutense de Madrid

Yu Kawamata
Kyoto University

Albano Galan
Institute of Chemical Research of Catalonia

Jochen Zoller
UpSolution Team
RWTH Aachen University

Fei Ji
Nanjing University of Science and Technology

Yoshinori Aihara
Osaka University

Sara Gutiérrez Hernández
University of Alcalá

Bala'zs Budai
École Polytechnique Fédérale de Lausanne

Iago Alonso Vicente
University of Vigo

Nathan Ferrandin
University Pierre & Marie Curie, Paris

Kasper Fjelbye
University of Copenhagen

Alex Novak
LMU Munich

Frederik Sandfort
University of Muenster

Lukas Nattmann
University of Muenster

Julien Vantourout
GSK–University of Strathclyde

Luca Buzzetti
ICIQ

Lucas Gottemann
LMU Munich

Monika Kruszyk
University of Copenhagen

Iñaki Bastida
University of the Basque Country (UPV/EHU)

Pedro Martín-Acosta
University Of La Laguna (IUBO-AG)

Cian Kingston
University College Dublin

Amin Minakar
University of Cologne

Sebastian Beil
Johannes Gutenberg University Mainz

Alberto Garrido-Castro
Universidad Autónoma de Madrid, Spain

Kosuke Yasui
Osaka University

Juan Miguel Lopez Soria
Instituto de Productos Naturales y Agrobiologia

Paula Fernández Canelas
University of Oviedo

Shengyang Ni
Nanjing University

Mauro Mato Gomez
ICIQ (Institute of Chemical Research of Catalonia)

Michal Ociepa
Institute of Organic Chemistry of the Polish Academy of Science

Alexander Sandahl
Aarhus University

Nazaret Rivas Bascón
University of Granada

Eva Rivera Chao
University of Santiago

Tao Sheng
Nanjing Agriculture University

Karolina Kowalska
University of Copenhagen
Adam Mickiewicz University
Adam Mickiewicz University

Yuxuan Chang
Nankai University

Edgar Molle
Karlsruhe Institute of Technology

Henrik Wilke
Ludwig-Maximilians-Universität Munchen

Simon Kolb
Technical University of Braunschweig

Sara
ICIQ

Laura Levy
CPE Lyon

Melania Prado Merini
Ruhr-Universität Bochum

Benedikt Nissl
LMU Munich
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Michael Giambrone
Cornell University

Brady Worrell
Purdue University

Ming Yan
Lafayette College

Cecil Eprile
Cornell University

Chao Wang
Lafayette College

Benjamin Winer
Diablo Valley College

Zachary Sweeney
Centre College

Brandon Whitefield
University of California San Diego

Leah Simke
University of Michigan

Adam Sobel

Steven Nguyen
University of California San Diego

Jonathan Nelson
University of California, San Diego

Joe Nagamizo
University of California, San Diego

Alex Nanna
Albion College

Soniya Gunjikar
University Institute of Chemical Technology, India

Rohan Merchant
University College London

Matt Del Bel
University of California, San Diego

Ryan Gianatassio
UMass–Boston

Angela Bai
University of California, San Diego

Sylvia Chen
University of Wisconsin-Madison

Garrett Michael Saul
University of California, San Diego

Lily Moloney
Augsburg College

Bryan J. Lee
University of California, San Diego

Kevin Nguyen
University of California, San Diego

Matthew ONeill
Notre Dame

Qian Zhenghao
University of Science and Technology of China

Cheng Bi
Nankai University

Yutong Lin
Nankai University

Brendyn Smith
Michigan State University

Jered Vaichis
University of California Irvine

Katarzyna Maziarz
Mount Holyoke College

Haolin Zhang
Tsinghua University

Zeyi ``Tony`` Huang
Nankai University

Fengyuan Wang
Tsinghua University

Miao Chen
Nankai University

Yunyeong Gwon
Daegu Gyeongbuk Institute of Science and Technology

Rohan Narayan
University of Delaware

Yuan Yuan
Peking University

Yuxuan Chang
Nankai University
High School Students

Lazer Shelley
Kearny High School

Jason Ge
UpSolution Team
Westview High School

Derek Barbas
Torrey Pines High School

Marcus Bray
UpSolution Team
Torrey Pines High School

Jacob Zhong
John P. Stevens High School

Antony Yu
Torrey Pines High School

Anish Velaparthi
West Windsor Plainsboro High School North